Cinitapride

Title: Cinitapride
CAS Registry Number: 66564-14-5
CAS Name: 4-Amino-N-[1-(3-cyclohexen-1-ylmethyl)-4-piperidinyl]-2-ethoxy-5-nitrobenzamide
Molecular Formula: C21H30N4O4
Molecular Weight: 402.49
Percent Composition: C 62.67%, H 7.51%, N 13.92%, O 15.90%
Literature References: Prepn: A. Vega-Noverola et al., DE 2751139 (1978 to Anphar); eidem, US 5026858 (1991 to Walton). Pharmacology: R. Massingham et al., J. Auton. Pharmacol. 5, 41 (1985). Spectral determn in pharmaceutical prepns: M. Blanco et al., J. Pharm. Sci. 82, 834 (1993). Clinical evaluation in functional dyspepsia, in comparison with metoclopramide, q.v.: F. Mora et al., Ann. Med. Interne 10, 323 (1993).
Derivative Type: Tartrate
CAS Registry Number: 96623-56-2
Manufacturers' Codes: LAS-17177
Trademarks: Cidine (Almirall)
Therap-Cat: Gastroprokinetic.
Keywords: Gastroprokinetic.
Cinmetacin Cinmethylin Cinnabarine Cinnamaldehyde Cinnamedrine

Cinitapride
Cinitapride.png
3D Cinitapride.png
Systematic (IUPAC) name
(RS)-4-amino-N-[1-(1-cyclohex-3-enylmethyl)-4-piperidyl]-2-ethoxy-5-nitro-benzamide
Clinical data
Legal status Prescription only
Routes Oral
Identifiers
CAS number 66564-14-5 YesY
ATC code None
PubChem CID 68867
DrugBank DB08810
ChemSpider 62099 YesY
UNII R8I97I2L24 YesY
KEGG D07700 YesY
Chemical data
Formula C21H30N4O4 
Mol. mass 402.49 g/mol
 YesY (what is this?)  (verify)

Cinitapride (Cintapro, Pemix) is a gastroprokinetic agent and antiulcer agent of the benzamide class which is marketed in India, Mexico, Pakistan and Spain.[1][2] It acts as an agonist of the 5-HT1 and 5-HT4 receptors and as an antagonist of the 5-HT2 receptors.[3][4]